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. Author manuscript; available in PMC: 2021 Jul 16.
Published in final edited form as: J Med Chem. 2021 Feb 1;64(3):1570–1583. doi: 10.1021/acs.jmedchem.0c01537

Table 1.

Growth Inhibitory Effects of the Four Compounds in GBM Cells

IC50 (nM)
compounds T98G U251 A172 U87
I 2.01 ± 0.64 4.00 ± 1.20 6.24 ± 1.06 4.78 ± 1.62
II 4.87 ± 2.04 6.39 ± 1.94 11.96 ± 2.77 6.74 ± 2.73
III 1.85 ± 0.81 1.57 ± 0.33 3.13 ± 0.78 3.05 ± 1.16
IV 5.71 ± 1.99 6.97 ± 1.08 8.21 ± 2.26 7.83 ± 3.81