Table 1.
NTMT1 inhibition evaluation of bisubstrate analogues
 | |||
|---|---|---|---|
| Compound ID | Peptide | n | Ki, app (nM) |
| 1 (NAH-C3-GPKK) | GPKK | 3 | 7 ± 1 |
| 2 (NAH-C4-GPKK) | GPKK | 4 | 5.0 ± 0.3 |
| 3 (NAH-C3-GPK) | GPK | 3 | 41 ± 4 |
| 4 (NAH-C4-GPK) | GPK | 4 | 44 ± 3 |
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