Table 4. C–H Iodination of Small-molecule Drugs^g.

^aReaction was conducted in 0.2 M MeCN.

^bReaction was conducted in 0.2 M DCM.

^cI₂ (1.3 equiv) and AgX (1.3 equiv).

^dLi₂CO₃ (1.0 equiv) was used.

^eI₂ (1.2 equiv) and AgOTf (1.2 equiv).

^fI₂ (1.5 equiv) and AgOTs (1.5 equiv).

^gGeneral conditions except where otherwise noted: arene (0.2 mmol), AgX (0.2 mmol, 1.0 equiv), I₂ (0.2 mmol, 1.0 equiv), 23 °C.