Table 1.
List of reference compounds used as agonists for the human TAS2R receptors in vitro assays.
| Receptor | Compound | Concentration |
|---|---|---|
| TAS2R1 | Oxyphenonium bromide | 3 mM |
| TAS2R3 | Chloroquine | 10 mM |
| TAS2R4 | Colchicine | 1 mM |
| TAS2R5 | 1,10-phenanthroline | 600 μM |
| TAS2R7 | Aurintrincarboxylic acid | 30 μM |
| TAS2R8 | Chloramphenicol | 300 μM |
| TAS2R9 | Ofloxacin | 3 mM |
| TAS2R10 | Oxyphenonium bromide | 3 mM |
| TAS2R13 | Denatonium benzoate | 3 mM |
| TAS2R14 | Aristolochic acid | 30 μM |
| TAS2R16 | Salicin | 3 mM |
| TAS2R20 | Ritanserin | 30 μM |
| TAS2R30 | Amarogentin | 10 μM |
| TAS2R31 | Aristolochic acid | 30 μM |
| TAS2R38 | Sinigrin | 3 mM |
| TAS2R39 | Denatonium benzoate | 3 mM |
| TAS2R40 | Cinchonine | 100 μM |
| TAS2R43 | Aristolochic acid | 30 μM |
| TAS2R46 | Strychnine | 10 μM |
| TAS2R50 | Andrographolide | 30 μM |
The reported concentrations are the highest used for each receptor.