Table 2.
Calculated values of Lipinski descriptors.
MW | LogP | NumH donors | NumH acceptors |
---|---|---|---|
281.3 | 1.90 | 0.0 | 5.0 |
416.5 | 3.82 | 0.0 | 2.0 |
422.2 | 2.67 | 0.0 | 3.0 |
294.3 | 3.63 | 0.0 | 4.0 |
339.3 | 3.54 | 0.0 | 5.0 |
338.4 | 3.41 | 0.0 | 5.0 |
297.0 | 3.45 | 0.0 | 3.0 |
277.2 | 4.10 | 0.0 | 3.0 |
278.3 | 3.30 | 0.0 | 3.0 |
282.4 | 4.11 | 0.0 | 2.0 |