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. 2021 Jul 12;13(14):3488. doi: 10.3390/cancers13143488

Table 1.

Efficacy and microsomal stability of the active AR-NTD inhibitors.

graphic file with name cancers-13-03488-i001.jpg

VPCID R1 R2 R4 R5 R6 R8 eGFP IC50 (μM) PSA IC50 (μM) PC3-iV7 IC50 (μM) T1/2 (min.)
220009 graphic file with name cancers-13-03488-i001.jpg graphic file with name cancers-13-03488-i002.jpg 1 1 NA
220010 graphic file with name cancers-13-03488-i003.jpg graphic file with name cancers-13-03488-i004.jpg 0.5 0.7 2.3 30
220027 graphic file with name cancers-13-03488-i005.jpg Br graphic file with name cancers-13-03488-i006.jpg Br 3 4 4 TBD
220028 graphic file with name cancers-13-03488-i007.jpg Br graphic file with name cancers-13-03488-i008.jpg Br 0.4 0.4 3 NA
220054 graphic file with name cancers-13-03488-i009.jpg graphic file with name cancers-13-03488-i010.jpg graphic file with name cancers-13-03488-i011.jpg 5 5 3 NA
220057 graphic file with name cancers-13-03488-i012.jpg graphic file with name cancers-13-03488-i013.jpg graphic file with name cancers-13-03488-i014.jpg graphic file with name cancers-13-03488-i015.jpg 10 8 8 462
220062 graphic file with name cancers-13-03488-i016.jpg Br graphic file with name cancers-13-03488-i017.jpg 0.5 0.5 3 36
220075 graphic file with name cancers-13-03488-i018.jpg graphic file with name cancers-13-03488-i019.jpg 0.5 0.5 12 18
RR-220010 graphic file with name cancers-13-03488-i020.jpg graphic file with name cancers-13-03488-i021.jpg 0.7 0.7 5 11
SS-220010 graphic file with name cancers-13-03488-i022.jpg graphic file with name cancers-13-03488-i023.jpg 0.7 0.6 6 12
RS-220010 graphic file with name cancers-13-03488-i024.jpg graphic file with name cancers-13-03488-i025.jpg 0.85 0.79 5 15