Table 2.
Kinetic parameters of PTP1B with different inhibitors.
| Compound | Ki (µM) | Inhibition Type |
|---|---|---|
| 4f | 3.9 ± 0.5 | non-competitive |
| 5f | 4.6 ± 0.6 | non-competitive |
| UA | 8.9 ± 0.7 | non-competitive |
| CL | 15.4 ± 1.7 | non-competitive |
| SU | 7.1 ± 0.9 | competitive |
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