Table 2.
Entry | Regents and conditions | Acid (equiv.) | 11b:11aa | Yields (%)b |
---|---|---|---|---|
1 | MeOH/CH3SO2OH, rt, 18 h | 5.5 | 1:0.66 | 32 |
2 | MeOH/HCl, rt, 3 h | 0.87 | 1:0.90 | 47 |
Ratio of 5-O-benzoyl β/α -xylofuranosides 11b and 11a determined from the 1H NMR spectrum of the anomeric mixture after treatment.
Yields of methyl 5-O-benzoyl α-xylofuranoside 11a refer to NMR yields.