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. Author manuscript; available in PMC: 2022 Apr 22.
Published in final edited form as: J Med Chem. 2021 Mar 31;64(8):5099–5122. doi: 10.1021/acs.jmedchem.1c00164

Figure 2.

Figure 2.

Inhibition of binding of fluorescent antagonist 2 at hP2Y14R (A) and at mP2Y14R (B) by four novel P2Y14R antagonist analogues (mean ± SD, n = 3–4 independent determinations, performed in triplicate).