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. 2021 Jul 14;12:667753. doi: 10.3389/fphar.2021.667753

TABLE 1.

Characteristics of Urate transporters.

Transporter Location in kidney Mutation Function of transporters
SLC2A9 (GLUT9) Apical and basolateral membranes of the renal proximal tubule R198W, R380C, P412R Anzai et al. (2008); Dinour et al. (2010); Kawamura et al. (2011) Urate reabsorption
SLC16A9 (MCT9) In the kidney and adrenal gland rs1171614 Butler et al. (2021) Related to UA levels
rs2242206 Nakayama et al. (2013)
SLC17A1 (NPT1) Apical membrane of the renal proximal tubule rs1165196 Chiba et al. (2015); Sakiyama et al. (2016) Urate absorption and efflux
I269T Sakiyama et al. (2016)
SLC17A3 (NPT4) Apical side of renal tubules rs9393672 Sakiyama et al. (2016); Jutabha et al. (2010); Riches et al. (2009) Urate excretion
rs942379 Sakiyama et al. (2016); Jutabha et al. (2010); Riches et al. (2009)
SLC22A6 (OAT1) Basolateral side of the proximal tubule ---- Urate excretion
SLC22A7 (OAT2) Mainly distributed in the kidney C329T, G571A, G1520A Xu et al. (2005); Kato et al. (2015) Urate secretion
SLC22A8 (OAT3) In the basolateral side of the proximal tubule ---- Urate excretion
SLC22A11 (OAT4) Proximal tubules of the kidney and other marginal epithelia rs2078267 Kenny et al. (2011); Flynn et al. (2013) Urate reabsorption
rs2186571 Kenny et al. (2011); Flynn et al. (2013)
rs17299124 Sakiyama et al. (2014)
rs17300741 Sakiyama et al. (2014)
SLC22A12 (URAT1) Apical membrane of the proximal tubule rs475688 Pavelcova et al. (2021) Urate reabsorption
ABCG2 Renal tubules and mesentery V12M, Q126X, Q141K, G268R, S441N, and F506SfsX4 Matsuo et al. (2009) Urate excretion
PDZK1 Apical membrane of the kidney proximal tubule rs12129861 Butler et al. (2021) Regulate the transport and activity of various transport proteins in the proximal tubules