Table-4. Ingredients for Dimenhydrinate ODTs with Superdisintegrant Bases.
|
Ingredients
(mg) |
Formulations | ||||||||||||
| F 1 | F 2 | F 3 | F 4 | F 5 | F 6 | F 7 | F 8 | F 9 | F 10 | F 11 | F 12 | F 13 | |
| Dimenhyrinate | 25 | 25 | 25 | 25 | 25 | 25 | 25 | 25 | 25 | 25 | 25 | 25 | 25 |
| SSG | 3 | 3 | 3 | 3 | 7.5 | 7.5 | 7.5 | 7.5 | 7.5 | 12 | 12 | 12 | 12 |
| CCS | 7 | 3.5 | 5.25 | 5.25 | 7 | 7 | 3.5 | 5.25 | 3.5 | 5.25 | 5.25 | 7 | 3.5 |
| CP | 5.25 | 5.25 | 3 | 7.5 | 3 | 7.5 | 3 | 5.25 | 7.5 | 7.5 | 3 | 5.25 | 5.25 |
| MCC | 30 | 30 | 30 | 30 | 30 | 30 | 30 | 30 | 30 | 30 | 30 | 30 | 30 |
| Sucralose | 5 | 5 | 5 | 5 | 5 | 5 | 5 | 5 | 5 | 5 | 5 | 5 | 5 |
| Mannitol | 72.75 | 76.25 | 76.75 | 72.25 | 70.5 | 66 | 74 | 70 | 69.5 | 63.25 | 67.75 | 63.75 | 65 |
| Mg stearate | 2 | 2 | 2 | 2 | 2 | 2 | 2 | 2 | 2 | 2 | 2 | 2 | 2 |
| Total weight | 150 | 150 | 150 | 150 | 150 | 150 | 150 | 150 | 150 | 150 | 150 | 150 | 150 |
SSG: Sodium starch glycolate; CCS: Croscarmellose sodium; CP: Crospovidone; MCC: Microcrystalline cellulose