Table 2.

List of pre-clinical direct MYC inhibitors

Mechanism	Type	Compound	References
Inhibitor of MYC/Max dimerization	Small Molecule	IIA6B17	[672]
		10058-F4	[673]
		10074-G5	[674]
		JY-3-094	[675]
		3jc48–3	[676]
		MYCro1, MYCro2, MYCro3	[677]
		MYCMI-6	[676]
		KJ-Pyr-9	[678]
		EN4	[679]
		MYCi361	[680]
		MYCi975	[681]
		KI-MS2-008	[682]
	(Poly)peptide	OmoMYC	[683]
		FPPa-OmoMYC	[684]
		Max bHLHZ (OmoMYC)	[685]
		Mxd1	[686]
		Monoclonal antibody	[687]
		H1 peptide	[688]
Inhibitor of E-box binding	Small Molecule	JKY-2-169	[689]
	(Poly)peptide	OmoMYC	[683]
		Max bHLHZ	[685]
		Mxd1	[686]
		ME47	[690]