Table 1.
Measured molecular masses of the protein species, including ternary complexes, detected from 9 μM Brd4B1 or Brd4B2, 9 μM VCB and 7.8 μM GNE‐987.
|
Brd4 Bromodomain |
Measured MW [Da] |
Corresponding Species |
Expected MW [Da] |
|---|---|---|---|
|
Brd4B1 |
18814.0 |
Apo‐Brd4B1 |
18814.4 |
|
19040.0 |
Biotinylated Apo‐Brd4B1 |
||
|
19911.7 |
Holo‐Brd4B1 |
19910.7 |
|
|
20135.6 |
Biotinylated Holo‐Brd4B1 |
||
|
45412.9 |
Holo‐VCB |
45412.7 |
|
|
64229.7 |
Ternary complex |
64227.1 |
|
|
64455.5 |
Ternary complex containing biotinylated Brd4B1 |
||
|
Brd4B2 |
17386.9 |
Apo‐Brd4B2 |
17386.8 |
|
18482.4 |
Holo‐Brd4B2 |
18483.1 |
|
|
44317.2 |
Apo‐VCB |
44316.4 |
|
|
45413.0 |
Holo‐VCB |
45412.7 |
|
|
62799.4 |
Ternary complex |
62799.5 |