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. 2021 Jun 23;14(14):2785–2853. doi: 10.1002/cssc.202100573

Scheme 5.

Scheme 5

Synthesis of 2 d (HBTU= 3‐[Bis(dimethylamino)methyliumyl]‐3H‐benzotriazol‐1‐oxide hexafluorophosphate, DIPEA= N,N‐diisopropylethylamine).