Scheme 5.

Synthesis of 2 d (HBTU= 3‐[Bis(dimethylamino)methyliumyl]‐3H‐benzotriazol‐1‐oxide hexafluorophosphate, DIPEA= N,N‐diisopropylethylamine).

Synthesis of 2 d (HBTU= 3‐[Bis(dimethylamino)methyliumyl]‐3H‐benzotriazol‐1‐oxide hexafluorophosphate, DIPEA= N,N‐diisopropylethylamine).