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. 2021 Aug 3;12(8):1308–1317. doi: 10.1021/acsmedchemlett.1c00294

Table 3. Full Curve BROMOscan Profiling of Compound 23a.

bromodomain compd 23 pKi
TAF1(2) 9.1
BRD4(1) <5.3 (>×6310)
BRD4(2) 6.1 (×1000)
BAZ2B 6.0 (×1260)
BRD9 7.4 (×50)
CECR2 6.0 (×1260)
BRPF1 5.3 (×6310)
a

TAF1(2) fold selectivity is shown in parentheses after the pKi value.