The IC50 for selected compounds which inhibit ADP-induced platelet aggregationa.
Compd | IC50 (μM) | Compd | IC50 (μM) |
---|---|---|---|
Ia | 4.89 | IIg | 0.67 |
Ic | 3.16 | IIh | 0.20 |
In | 1.78 | IIi | 0.78 |
Io | 0.82 | IIl | 1.30 |
IIe | 0.58 | IIr | 0.66 |
IIf | 0.45 | IIu | 0.40 |
Ticagrelor | 0.74 |
ADP-induced platelet aggregation ([ADP] = 10 μM).