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. 2021 Jul 13;12(8):1414–1427. doi: 10.1039/d1md00128k

The IC50 for selected compounds which inhibit ADP-induced platelet aggregationa.

Compd IC50 (μM) Compd IC50 (μM)
Ia 4.89 IIg 0.67
Ic 3.16 IIh 0.20
In 1.78 IIi 0.78
Io 0.82 IIl 1.30
IIe 0.58 IIr 0.66
IIf 0.45 IIu 0.40
Ticagrelor 0.74
a

ADP-induced platelet aggregation ([ADP] = 10 μM).