Chemical and metabolic stability of compound IIh.
Assay | IIh | |
---|---|---|
Chemical stability | PBS, 37 °C, 1 week | 98.3% |
FaSSGF, 1 day | 96.7% | |
FaSSIF, 1 day | 97.4% | |
Metabolic stability (MLM, remaining) | 1 h | 81.2% |
2 h | 73.7% |
Assay | IIh | |
---|---|---|
Chemical stability | PBS, 37 °C, 1 week | 98.3% |
FaSSGF, 1 day | 96.7% | |
FaSSIF, 1 day | 97.4% | |
Metabolic stability (MLM, remaining) | 1 h | 81.2% |
2 h | 73.7% |