Chemical and metabolic stability of compound IIh.
| Assay | IIh | |
|---|---|---|
| Chemical stability | PBS, 37 °C, 1 week | 98.3% |
| FaSSGF, 1 day | 96.7% | |
| FaSSIF, 1 day | 97.4% | |
| Metabolic stability (MLM, remaining) | 1 h | 81.2% |
| 2 h | 73.7% | |
| Assay | IIh | |
|---|---|---|
| Chemical stability | PBS, 37 °C, 1 week | 98.3% |
| FaSSGF, 1 day | 96.7% | |
| FaSSIF, 1 day | 97.4% | |
| Metabolic stability (MLM, remaining) | 1 h | 81.2% |
| 2 h | 73.7% | |