Table 3.
The AUC ratio and Cmax ratio of the DDI profiles for PO OXY and 10 mg, 100 mg, 500 mg and 1000 mg of PO DZP when applying mixed-type inhibition to the DDI model. CI is the 95% Confidence Interval. AUC24h ratio is the exposure of AUC ratio from the time 0 to 24 hours.
| Dosing Strategy | AUC24h ratio | CI [5%,95%] | Cmax ratio | CI [5%,95%] |
|---|---|---|---|---|
| OXY 30 mg + DZP 10mg | 1.01 | [1.01,1.02] | 1.01 | [1.00,1.02] |
| OXY 30 mg + DZP 100mg | 1.07 | [1.04,1.09] | 1.04 | [1.03,1.06] |
| OXY 30 mg + DZP 500mg | 1.21 | [1.13,1.31] | 1.10 | [1.06,1.16] |
| OXY 30 mg + DZP 1000mg | 1.30 | [1.17,1.48] | 1.13 | [1.07,1.22] |