Table 3.
Mouse plasma and liver trough levels 24 h after 3rd 100 mg/kg dose
| Compound | Plasma (μM)a | Liver (μM)a | ||
|---|---|---|---|---|
| Male | Female | Male | Female | |
| ARN-75039 | 21.1 ± 5.5 | 22.1 ± 14.1 | 71.8 ± 19.4 | 79.2 ± 66.0 |
| ARN-75041 | 10.8b | 21.2b | 150.0 ± 15.1 | >200c |
Data points represent the mean and standard deviation of 3 mice per sex
Plasma samples pooled from 3 mice
Measured concentration above the upper limit of the standard curve