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. 2021 Aug 10;8:702776. doi: 10.3389/fmed.2021.702776

Table 2.

Summary of the demographic data of patients enrolled in clinical trials testing the efficacy of IL-23, IL-23/12, IL-17, IL-17RA, and TNF-α inhibitors.

References Phase Biologic Dosing scheme Endpoint week Total (n) Age (years) Male (%) Weight (kg) BMI (kg/m ∧ 2) Disease duration (years) % body surface
Resurface 1 (103) (dosing scheme summary only from part 1) 3 Tildrakizumab 100 mg, week 0, 4 12 309 46.4 67 88.5 29.7
Tildrakizumab 200 mg, week 0, 4 12 308 46.9 73 88.9 30.9
Placebo 12 154 47.9 65 87.5 29.6
Resurface 2 (103) (dosing scheme summary only from part 1) 3 Tildrakizumab 100 mg, week 0, 4 12 307 44.6 72 89.4 34.2
Tildrakizumab 200 mg, week 0, 4 12 314 44.6 72 88.4 31.8
Etanercept 50 mg, week 0, 4 12 313 45.8 71 88 31.6
Placebo 12 156 46.4 72 88.7 31.3
Papp et al. (102) 2b Tildrakizumab 5 mg, week 0, 4 12 42 43.2 74 28.9
Tildrakizumab 25 mg week 0, 4 12 92 46.3 65 28.5
Tildrakizumab 100 mg week 0.4 12 89 45.5 85 29
Tildrakizumab 200 mg week 0, 4 12 86 43.2 76 28.5
Placebo 12 46 45.9 83 29.5
Kopp et al. (101) 1 Tildrakizumab 3 mg/kg–weeks 0, 4 28 7 52.7 100 90.27
Tildrakizumab 10 mg/kg–weeks 0, 4 28 6 46.2 67 94.25
Placebo 28 20 45.5 80 102.46
Voyage 1 (72) 3 Guselkumab 100 mg–week 0, 4 16 329 43.9 72.9 29.7 17.9 28.3
Placebo 16 174 44.9 68.4 28.9 17.6 25.8
Voyage 2 (74) 3 Guselkumab 100 mg–week 0, 4 16 496 43.7 70.4 29.6 17.9 28.5
Placebo 16 248 43.3 69.8 29.6 17.9 28
UltIMMa-1 (79) 3 Risankizumab 150 mg–week 0, 4 16 304 48.3 70 87.8 26.2
Placebo 16 102 49.3 77 88.8 27.9
UltIMMa-2 (79) 3 Risankizumab 150 mg–week 0, 4 16 294 46.2 69 92.2 26.2
Placebo 16 98 46.3 68 92.2 23.9
Reich et al. (82) 2 Mirikizumab 100 mg–week 0, 8 16 51 46 69 86.4 18.6 26.5
Mirikizumab 300 mg–week 0, 8 16 51 47.5 71 87.9 18.1 21.3
Placebo 16 52 46 81 89.1 18 26.4
Phoenix-1 (51) 3 Ustekinumab 90 mg–week 0, 4 12 256 46.2 67.6 93.8 19.6 25.2
Placebo 12 255 44.8 71.8 94.2 20.4 27.7
Phoenix-2 (52) 3 Ustekinumab 90 mg–week 0, 4 12 411 46.6 66.7 91.5 20.3 27.1
Placebo 12 410 47 69 91.1 20.8 26.1
FIXTURE (135) 3 Secukinumab 150 mg–weeks 0–4 then every 4 weeks thereafter 12 327 45.4 72.2 83.6 17.3 34.5
Secukinumab 300 mg–weeks 0–4 then every 4 weeks thereafter 12 327 44.5 68.5 83 15.8 34.3
Placebo 12 326 44.1 72.7 82 16.6 35.2
Etanercept 50 mg–weeks 0–4 then every 4 weeks thereafter 12 326 43.8 71.2 84.6 16.4 33.6
UNCOVER-1 (123) 3 Ixekizumab 160 mg × 1, 80 mg (q2w) 12 433 45 67.2 92 20 27
Ixekizumab 160 mg × 1, 80 mg (q4w) 12 432 46 66.9 92 19 28
Placebo 12 431 46 70.3 92 20 27
AMAGINE-1 (136) 3 Brodalumab 140 mg q2w 12 219 46 74 90.6 19 27.4
Brodalumab 210 mg q2w 12 222 46 73 91.4 20 25.1
Placebo 12 220 47 73 90.4 21 26.9
BE ABLE 1 (137) 2b Bimekizumab 160 mg q4w 12 40 43.4 65.1 91.6 15.9 24
Bimekizumab 320 mg q4w 12 43 42.6 74.4 86.9 15.9 24
Placebo 12 42 46.7 59.5 88.8 15 25.5
EXPRESS II (138) Infliximab 5 mg/kg 14 314 44.5 65 92.2 19.1 28.7
Placebo 14 208 44.4 69.2 91.1 17.8 28.4
REVEAL (139) 3 Adalimumab 40 mg q2w 15 814 44.1 67.1 92.3 18.1 25.8
Placebo 15 398 45.4 64.6 94.1 18.4 25.6
CIMPACT (140) 3 Certolizumab pegol 200 mg q2w 16 165 46.7 68.5 89.7 19.5 28.1
Placebo 16 57 46.5 59.6 93.7 18.9 24.3
GO-VIBRANT (141) 3 Golimumab 2 mg/kg, weeks 0, 4 then every 8 weeks thereafter 16 241 45.7 53.1 6.2
Placebo 16 239 46.7 50.6 5.3