Fig. 3.
Specificity of the DYRK1A harmine-related alkaloid inhibitors against a kinase panel. (A) To assess selectivity, compounds (at 10 μM) were profiled for selectivity against a panel of 10 kinases (Reaction Biology Corp., n = 2). Reductions in enzyme activity (%) are shown for each compound as a separate bar chart. (B) Human kinome map highlighting CMGC family with eight of the kinase selectivity panel highlighted by black circles and DYRK1A by a red circle. Human Kinome illustration reproduced courtesy of Cell Signaling Technology, Inc. (www.cellsignal.com).