Table 2.
Effect of inhibitors on ginger polyphenol oxidase. Km, Vmax, Ki and I50 values were shown
Inhibitors | [I] (mg/mL) | I50 (mg/mL) | Inhibition (%) | Vmax (EU/min/mL) | Km (mM) | Ki (mM) | Type of inhibition |
---|---|---|---|---|---|---|---|
Control Sonneratia.alba |
25,241.12 | 3.29 | |||||
0.125 | 1.013 | 24.88 | 17,420.45 | 3.28 | 0.28 | Non-competitive | |
0.25 | 34.27 | 15,994.98 | 3.24 | 0.43 | |||
0.5 | 35.68 | 15,305.64 | 3.28 | 0.77 | |||
Rhizophora apiculate | 0.125 | 0.672 | 23.47 | 18,570.31 | 4.31 | 0.35/1.78 | Mixed |
0.25 | 39.44 | 15,392.52 | 4.72 | 0.39/2.35 | |||
0.5 | 40.85 | 15,038.48 | 5.02 | 0.74/2.56 | |||
Syzygium grande | 0.125 | 1.005 | 32.39 | 17,515.04 | 2.45 | 0.28 | Un-competitive |
0.25 | 35.21 | 15,740.07 | 2.16 | 0.41 | |||
0.5 | 39.91 | 15,106.13 | 2.08 | 0.75 | |||
Rhizophora mucronata | 0.125 | 0.535 | 15.49 | 21,311.33 | 2.95 | 0.68 | Un-competitive |
0.25 | 41.31 | 14,656.42 | 2.16 | 0.35 | |||
0.5 | 44.13 | 13,864.16 | 2.03 | 0.61 | |||
Hibiscus tiliaceus | 0.125 | 0.560 | 14.55 | 21,418.46 | 3.49 | 0.70/1.25 | Mixed |
0.25 | 36.62 | 15,393.00 | 3.81 | 0.39/1.90 | |||
0.5 | 43.19 | 14,328.29 | 3.91 | 0.66/2.09 | |||
Bruguiera gymnorhiza | 0.125 | 0.527 | 10.80 | 22,194.50 | 2.86 | 0.91 | Un-competitive |
0.25 | 39.44 | 14,570.95 | 1.86 | 0.34 | |||
0.5 | 44.13 | 13,523.47 | 1.70 | 0.58 |