Table 1.
Compound | Ki [nM] ± SEM | ||
---|---|---|---|
MOR | DOR | KOR | |
Dmt-DALDA | 0.61 ± 0.02 | 2313 | 128.98 ± 8.02 |
KGOP01 | 0.12 ± 0.06 | 4.88 ± 0.11 | 72.75 ± 4.32 |
SBL-OPNK-4 | 1.02 ± 0.03 | 1251.18 | 90.50 ± 5.69 |
SBL-OPNK-5 | 2.11 ± 0.04 | 10.02 ± 3.20 | 90.72 ± 0.94 |
SBL-OPNK-6 | 74.93 ± 0.15 | 22377 | 100.44 ± 1.16 |
SBL-OPNK-7 | 2.83 ± 0.02 | 3.26 ± 0.09 | 52.98 ± 3.20 |
SBL-OPNK-8 | 119.68 ± 5.25 | 4574.17 | 103.83 ± 6.12 |
SBL-OPNK-9 | 5.43 ± 0.08 | 6.57 ± 4.02 | 97.15 ± 4.72 |