Table 2. Physiochemical Properties and Brain-to-Plasma Ratios (AUCbrain/AUCplasma) of Anti-AβO Compounds.
| cmpd | MW | cLogP | tPSA | Brain/plasma AUC | Brain/plasma 24 h postdose |
|---|---|---|---|---|---|
| (R)-2 | 376.2 | 6.48 | 12.3 | NT | 8.2 |
| 3 | 341.8 | 5.89 | 12.0 | NT | 2.0 |
| 6 | 357.5 | 4.65 | 32.7 | 5.64 | 5.4 |
| 7 | 431.6 | 3.26 | 66.8 | 2.51 | 5.7 |