Table 3. Sensitivity of HIV-1BaL to PAPEG27 in TZM-bl Cells.
|
N-PA |
C-PA |
K-PA |
|||||||
|---|---|---|---|---|---|---|---|---|---|
| inhibitory conc.a | monoalkyl | dialkyl | chol | monoalkyl | dialkyl | chol | monoalkyl | dialkyl | chol |
| IC50 (μM) | 0.20 | 0.15 | 0.12 | 0.08 | N/A | 1.71 | 0.37 | 0.05 | 0.09 |
| (0.04) | (0.04) | (0.07) | (0.01) | (0.72) | (0.17) | (0.04) | (0.01) | ||
| IC95 (μM) | 5.87 | N/A | N/A | 5.60 | N/A | N/A | N/A | N/A | N/A |
| (0.72) | (0.93) | ||||||||
| SI (CC50/IC50) | 85 | - | - | 250 | - | - | - | - | - |
The IC values shown are the means (SEM) derived from the triplicates for each condition performed.