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. 2021 Jul 13;32(9):1999–2013. doi: 10.1021/acs.bioconjchem.1c00292

Table 3. Sensitivity of HIV-1BaL to PAPEG27 in TZM-bl Cells.

  N-PA
C-PA
K-PA
inhibitory conc.a monoalkyl dialkyl chol monoalkyl dialkyl chol monoalkyl dialkyl chol
IC50 (μM) 0.20 0.15 0.12 0.08 N/A 1.71 0.37 0.05 0.09
(0.04) (0.04) (0.07) (0.01)   (0.72) (0.17) (0.04) (0.01)
IC95 (μM) 5.87 N/A N/A 5.60 N/A N/A N/A N/A N/A
(0.72)     (0.93)          
SI (CC50/IC50) 85 - - 250 - - - - -
a

The IC values shown are the means (SEM) derived from the triplicates for each condition performed.