Table 4.
Metabolites | Structure | Km, µM | Vmax, pmol/min/mg microsomal protein | Catalytic efficiency (Vmax/Km), µl/min/mg protein |
---|---|---|---|---|
9,10-dihydro-B[a]P-diol | 11.9 ± 5.5 | 28.3 ± 2.8 | 2.4 | |
4,5-dihydro-B[a]P-diol | 6.5 ± 4.5 | 13.3 ± 1.4 | 2.0 | |
7,8-dihydro-B[a]P-diol | 14.6 ± 9.8 | 7.0 ± 1.1 | 0.5 | |
7,8-dihydro-B[a]P-diol | 12.6 ± 10.7 | 13.3 ± 2.5 | 1.1 | |
B[a]P-1,6-quinone | 14.8 ± 8.8 | 22.2 ± 3.2 | 1.5 | |
B[a]P-3,6-quinone | 24.0 ± 14.4 | 3.0 ± 0.5 | 0.1 | |
9-hydroxy-B[a]P | 11.4 ± 5.2 | 20.0 ± 1.9 | 1.8 | |
3-hydroxy-B[a]P | 34.2 ± 17.7 | 162.2 ± 47.6 | 7.8 |