Table 1.
Summary of individual NanoBRET(TM) Kinase assay components and expected assay outcomes using control inhibitors CC1 or crizotinib
| Kinase | Product # (promega) | Diluent DNA | Orientation of Nluc | [NanoBRET(TM) tracer K10], nM | BRET S:B (BRETTracer / BRETno tracer) | CC1 % occupancy, 300 nM | St dev | Crizotinib % occupancy, 1 uM | St dev |
|---|---|---|---|---|---|---|---|---|---|
| LRRK2 | NV340A | Transfection Carrier | C | 25 | 3.7 | 98 | 2.0 | −9 | 15.2 |
| MAPK6 | NV169A | Transfection Carrier | N | 25 | 7.4 | 99 | 0.8 | 2 | 2.4 |
| IRAK3 | NV144A | Transfection Carrier | N | 25 | 4.5 | 98 | 0.8 | 42 | 4.4 |
| TEK | NV215A | Transfection Carrier | C | 25 | 3.7 | 90 | 1.0 | 37 | 4.7 |
| TNK1 | NV218A | Transfection Carrier | N | 25 | 10.0 | 94 | 0.8 | −6 | 4.1 |
| GAK | NV142A | Transfection Carrier | N | 25 | 14.9 | 97 | 0.5 | −14 | 1.5 |
| MAPK4 | NV168A | Transfection Carrier | N | 25 | 26.8 | 97 | 1.2 | −12 | 3.4 |
| AAK1 | NV100A | Transfection Carrier | N | 25 | 12.2 | 99 | 0.3 | −14 | 0.9 |
| AURKA | NV104A | Transfection Carrier | C | 25 | 6.8 | 93 | 1.0 | 30 | 7.7 |
| AURKC | NV106A | Transfection Carrier | C | 25 | 10.6 | 92 | 1.8 | 48 | 4.2 |
| AURKB | NV105A | Transfection Carrier | C | 25 | 10.7 | 94 | 1.6 | 46 | 5.9 |
| NUAK1 | NV183A | Transfection Carrier | N | 25 | 3.4 | 98 | 2.4 | 36 | 6.6 |
| LATS2 | NV151A | Transfection Carrier | C | 25 | 5.0 | 79 | 7.1 | −10 | 6.2 |
| RPS6KA3 | NV200A | Transfection Carrier | N | 25 | 3.6 | 97 | 0.9 | −7 | 7.7 |
| SNF1LK2 | NV206A | Transfection Carrier | N | 25 | 16.9 | 99 | 0.5 | 0 | 3.4 |
| MYLK2 | NV177A | Transfection Carrier | C | 25 | 6.2 | 99 | 0.4 | −16 | 8.3 |
| AXL | NV107A | Transfection Carrier | C | 250 | 2.9 | 63 | 3.8 | 68 | 1.5 |
| FGFR3 | NV136A | Transfection Carrier | C | 250 | 3.4 | 84 | 4.1 | 14 | 6.8 |
| FLT3 | NV139A | Transfection Carrier | C | 250 | 3.4 | 79 | 3.7 | −4 | 8.6 |
| IGF1R | NV326A | Transfection Carrier | C | 250 | 2.1 | 78 | 3.8 | 18 | 8.2 |
| INSR | NV327A | Transfection Carrier | C | 250 | 2.9 | 83 | 2.5 | 20 | 2.1 |
| LIMK2 | NV153A | Transfection Carrier | C | 250 | 4.2 | 76 | 3.6 | 32 | 9.8 |
| TEC | NV214A | Transfection Carrier | N | 250 | 4.6 | 78 | 1.4 | −7 | 6.7 |
| TIE1 | NV217A | Transfection Carrier | C | 250 | 9.9 | 67 | 7.2 | 35 | 9.9 |
| CLK1 | NV113A | Transfection Carrier | N | 250 | 7.3 | 98 | 0.7 | 0 | 3.4 |
| SBK3 | NV421A | Transfection Carrier | N | 250 | 4.1 | 90 | 4.4 | 41 | 5.6 |
| NEK9 | NV180A | Transfection Carrier | N | 250 | 7.9 | 65 | 5.2 | 1 | 5.4 |
| NEK3 | NV179A | Transfection Carrier | N | 250 | 16.1 | 44 | 9.6 | −2 | 14.5 |
| NIM1K | NV381A | Transfection Carrier | C | 250 | 4.6 | 82 | 4.9 | −3 | 1.7 |
| STK36 | NV433A | Transfection Carrier | N | 250 | 7.1 | 89 | 3.8 | −6 | 6.5 |
| ULK2 | NV222A | Transfection Carrier | N | 250 | 10.5 | 78 | 8.0 | −1 | 1.9 |
| ULK3 | NV449A | Transfection Carrier | N | 250 | 23.1 | 72 | 5.2 | 2 | 6.5 |
| BRSK1 | NV249A | Transfection Carrier | N | 250 | 8.3 | 78 | 7.1 | −1 | 4.0 |
| MAP3K10 | NV156A | Transfection Carrier | N | 250 | 4.5 | 54 | 3.3 | −1 | 4.4 |
| MAP3K9 | NV160A | Transfection Carrier | N | 250 | 2.9 | 60 | 4.3 | −1 | 6.2 |
| MYLK3 | NV374A | Transfection Carrier | C | 250 | 8.5 | 72 | 9.1 | −8 | 6.4 |
| PHKG1 | NV186A | Transfection Carrier | N | 250 | 5.9 | 86 | 3.1 | −3 | 6.3 |
| STK33 | NV211A | Transfection Carrier | N | 250 | 3.1 | 90 | 3.4 | −3 | 3.9 |
| STK4 | NV435A | Transfection Carrier | N | 250 | 4.8 | 67 | 2.4 | 11 | 7.6 |
| TLK1 | NV443A | Transfection Carrier | C | 250 | 2.8 | 5 | 1.9 | −5 | 3.8 |
| FGFR1 | NV134A | Transfection Carrier | C | 100 | 3.3 | 95 | 1.8 | 0 | 3.8 |
| FGFR2 | NV135A | Transfection Carrier | C | 100 | 3.5 | 94 | 0.7 | 10 | 1.8 |
| MUSK | NV176A | Transfection Carrier | C | 100 | 3.3 | 89 | 4.3 | 80 | 2.8 |
| NTRK1 | NV181A | Transfection Carrier | C | 100 | 4.1 | 68 | 4.5 | 71 | 2.5 |
| RET | NV195A | Transfection Carrier | C | 100 | 6.0 | 90 | 1.5 | 4 | 4.5 |
| NTRK2 | NV182A | Transfection Carrier | C | 100 | 4.6 | 80 | 3.4 | 85 | 2.3 |
| TNK2 | NV445A | Transfection Carrier | C | 100 | 6.8 | 73 | 4.0 | 13 | 6.7 |
| LTK | NV154A | Transfection Carrier | C | 100 | 4.2 | 71 | 4.3 | 87 | 0.9 |
| BRAF(V600E) | NV248A | Transfection Carrier | C | 100 | 3.9 | 39 | 5.8 | −4 | 3.9 |
| IRAK4 | NV145A | Transfection Carrier | C | 100 | 6.5 | 98 | 1.4 | 6 | 7.0 |
| ITK | NV146A | Transfection Carrier | N | 100 | 3.4 | 92 | 1.8 | −1 | 6.2 |
| JAK2 (V617F) | NV330A | Transfection Carrier | C | 100 | 3.3 | 90 | 2.8 | 65 | 8.3 |
| MAP3K11 | NV157A | Transfection Carrier | N | 100 | 4.6 | 71 | 4.9 | 0 | 6.0 |
| PTK2 | NV192A | Transfection Carrier | N | 100 | 3.3 | 88 | 1.2 | 40 | 4.0 |
| PTK6 | NV194A | Transfection Carrier | C | 100 | 3.7 | 100 | 0.6 | −2 | 1.2 |
| PTK2B | NV193A | Transfection Carrier | C | 100 | 2.2 | 91 | 2.2 | 47 | 5.1 |
| BMP2K | NV109A | Transfection Carrier | N | 100 | 8.9 | 94 | 1.6 | 11 | 6.0 |
| NEK5 | NV379A | Transfection Carrier | N | 100 | 16.2 | 85 | 1.2 | −6 | 2.1 |
| STK16 | NV209A | Transfection Carrier | N | 100 | 13.4 | 85 | 1.9 | −13 | 6.2 |
| TBK1 | NV213A | Transfection Carrier | N | 100 | 7.5 | 78 | 4.2 | −7 | 10.8 |
| ULK1 | NV221A | Transfection Carrier | N | 100 | 14.2 | 94 | 1.9 | −1 | 5.5 |
| MAP4K2 | NV162A | Transfection Carrier | N | 100 | 4.5 | 76 | 2.0 | 77 | 10.7 |
| WEE1 | NV223A | Transfection Carrier | C | 100 | 5.3 | 91 | 1.0 | −9 | 2.5 |
| MYLK4 | NV375A | Transfection Carrier | C | 100 | 6.1 | 99 | 0.7 | −8 | 8.4 |
| MARK4 | NV173A | Transfection Carrier | N | 100 | 4.4 | 90 | 2.0 | −15 | 4.5 |
| PRKAA1 | NV410A | Transfection Carrier | N | 100 | 11.3 | 92 | 1.5 | −1 | 4.9 |
| PRKAA2 | NV189A | Transfection Carrier | N | 100 | 12.6 | 97 | 0.3 | −6 | 2.2 |
| RPS6KA1 | NV198A | Transfection Carrier | N | 100 | 7.9 | 89 | 1.9 | −6 | 2.5 |
| RPS6KA2 | NV199A | Transfection Carrier | N | 100 | 4.7 | 79 | 4.2 | −7 | 7.5 |
| RPS6KA4 | NV201A | Transfection Carrier | N | 100 | 6.6 | 85 | 0.7 | −11 | 6.0 |
| RPS6KA6 | NV202A | Transfection Carrier | N | 100 | 3.0 | 89 | 2.3 | −10 | 7.3 |
| SIK1 | NV203A | Transfection Carrier | N | 100 | 10.2 | 93 | 1.6 | −4 | 4.7 |
| CLK4 | NV115A | Transfection Carrier | C | 100 | 2.5 | 101 | 1.4 | −19 | 4.6 |
| MAPK8 | NV170A | Transfection Carrier | N | 100 | 5.8 | 70 | 7.8 | −16 | 4.2 |
| MAPK9 | NV171A | Transfection Carrier | N | 100 | 9.4 | 70 | 6.4 | −11 | 2.1 |
| IKBKE | NV143A | Transfection Carrier | N | 100 | 7.7 | 74 | 5.2 | 21 | 2.8 |
| LATS1 | NV150A | Transfection Carrier | C | 100 | 5.1 | 68 | 5.7 | −10 | 3.9 |
| PRKX | NV191A | Transfection Carrier | C | 100 | 3.6 | 65 | 4.9 | −14 | 7.9 |
| CSNK2A2 | NV119A | Transfection Carrier | C | 100 | 5.5 | 87 | 3.0 | −14 | 5.8 |
| HIPK4 | NV324A | Transfection Carrier | N | 100 | 7.8 | 97 | 0.4 | −9 | 6.1 |
| STK10 | NV426A | Transfection Carrier | C | 1000 | 2.8 | 80 | 3.4 | 35 | 3.0 |
| FGFR4 | NV137A | Transfection Carrier | C | 1000 | 3.5 | 68 | 4.0 | 3 | 1.6 |
| MAP4K1 | NV161A | Transfection Carrier | N | 1000 | 3.9 | 70 | 4.5 | 14 | 4.1 |
| MERTK | NV356A | Transfection Carrier | C | 1000 | 2.2 | 48 | 3.9 | 58 | 3.3 |
| MET | NV175A | Transfection Carrier | C | 1000 | 5.1 | 42 | 8.5 | 95 | 1.1 |
| RON | NV418A | Transfection Carrier | C | 1000 | 3.9 | 32 | 9.9 | 86 | 4.8 |
| TYRO3 | NV448A | Transfection Carrier | C | 1000 | 2.5 | 47 | 0.5 | 49 | 2.2 |
| LCK | NV152A | Transfection Carrier | C | 1000 | 3.8 | 78 | 4.2 | 36 | 5.7 |
| LIMK1 | NV339A | Transfection Carrier | C | 1000 | 5.2 | 69 | 5.6 | 29 | 5.5 |
| EPHA1 | NV122A | Transfection Carrier | C | 1000 | 3.3 | 74 | 3.2 | 75 | 2.2 |
| EPHA4 | NV124A | Transfection Carrier | C | 1000 | 2.8 | 33 | 5.2 | 53 | 4.4 |
| EPHA6 | NV126A | Transfection Carrier | C | 1000 | 3.9 | 38 | 1.7 | 64 | 5.1 |
| EPHA7 | NV127A | Transfection Carrier | C | 1000 | 4.4 | 51 | 4.6 | 38 | 2.4 |
| EPHB1 | NV307A | Transfection Carrier | C | 1000 | 3.4 | 65 | 2.4 | 68 | 2.0 |
| EPHB4 | NV131A | Transfection Carrier | C | 1000 | 3.1 | 53 | 4.9 | 62 | 3.6 |
| FYN | NV141A | Transfection Carrier | C | 1000 | 3.9 | 65 | 7.5 | −2 | 12.3 |
| ABL2 | NV233A | Transfection Carrier | N | 1000 | 2.9 | 72 | 5.5 | 43 | 3.9 |
| BMX | NV110A | Transfection Carrier | C | 1000 | 4.5 | 60 | 6.3 | 7 | 4.3 |
| BTK | N244A | Transfection Carrier | C | 1000 | 6.8 | 75 | 4.4 | 1 | 1.3 |
| FER | NV133A | Transfection Carrier | C | 1000 | 2.8 | 66 | 4.9 | 16 | 7.9 |
| FES | NV309A | Transfection Carrier | C | 1000 | 3.0 | 43 | 7.6 | 1 | 2.5 |
| JAK3 | NV147A | Transfection Carrier | C | 1000 | 4.7 | 45 | 4.8 | 2 | 4.4 |
| SRMS | NV425A | Transfection Carrier | N | 1000 | 2.7 | 18 | 4.3 | 0 | 4.9 |
| TXK | NV220A | Transfection Carrier | C | 1000 | 2.6 | 60 | 13.1 | 18 | 2.8 |
| CLK2 | NV114A | Transfection Carrier | C | 1000 | 4.1 | 89 | 2.2 | 1 | 4.7 |
| DYRK1A | NV303A | Transfection Carrier | N | 1000 | 2.6 | 78 | 4.4 | 0 | 5.3 |
| DYRK1B | NV121A | Transfection Carrier | N | 1000 | 3.3 | 87 | 3.6 | 0 | 2.1 |
| ERN1 | NV132A | Transfection Carrier | C | 1000 | 3.6 | 83 | 1.3 | −3 | 8.1 |
| ERN2 | NV308A | Transfection Carrier | C | 1000 | 5.3 | 61 | 7.4 | −9 | 13.9 |
| HIPK2 | NV322A | Transfection Carrier | N | 1000 | 3.3 | 82 | 2.8 | 5 | 4.4 |
| HIPK3 | NV323A | Transfection Carrier | N | 1000 | 1.9 | 70 | 14.3 | −4 | 14.6 |
| ICK | NV325A | Transfection Carrier | N | 1000 | 2.6 | 47 | 11.0 | 3 | 15.4 |
| CDK1 | NV270A | CycB1 (NV260A) | C | 1000 | 3.0 | 71 | 7.1 | 7 | 2.9 |
| CDK2 | NV278A | CycE1 (NV264A) | C | 1000 | 12.5 | 80 | 4.0 | 3 | 1.6 |
| CDK3 | NV280A | CycE1 (NV264A) | C | 1000 | 6.9 | 85 | 3.5 | 6 | 1.3 |
| CDK4 | NV281A | CycD3 (NV263A) | N | 1000 | 8.2 | 93 | 2.2 | 4 | 4.2 |
| CDK5 | NV112A | CDK5R1 (NV282A | C | 1000 | 13.3 | 85 | 3.6 | 1 | 0.8 |
| CDK6 | NV284A | CycD1 (NV262A) | N | 1000 | 4.1 | 89 | 2.2 | 0 | 3.0 |
| CDK7 | NV285A | Transfection Carrier | N | 1000 | 3.3 | 83 | 4.1 | 32 | 1.3 |
| CDK9 | NV287A | CycK (NV266A) | N | 1000 | 3.8 | 68 | 4.1 | 4 | 5.5 |
| CDK10 | NV271A | CycL2 (NV267A) | C | 1000 | 2.9 | 50 | 3.7 | 8 | 0.5 |
| CDK14 | NV272A | CycY (NV269A) | C | 1000 | 4.3 | 82 | 1.3 | 0 | 2.4 |
| CDK15 | NV273A | CycY (NV269A) | N | 1000 | 3.5 | 78 | 2.1 | 3 | 2.8 |
| CDK16 | NV274A | CycY (NV269A) | C | 1000 | 7.2 | 96 | 0.6 | 2 | 0.4 |
| CDK17 | NV275A | CycY (NV269A) | C | 1000 | 9.6 | 95 | 0.8 | 3 | 3.6 |
| CDK18 | NV276A | CycY (NV269A) | C | 1000 | 11.4 | 86 | 1.4 | 2 | 2.1 |
| CDKL2 | NV289A | Transfection Carrier | N | 1000 | 6.7 | 95 | 1.3 | 21 | 0.7 |
| CDK20 | NV279A | CycH (NV265A) | N | 1000 | 4.3 | 54 | 4.9 | −11 | 5.0 |
| CDKL1 | NV288A | Transfection Carrier | N | 1000 | 5.1 | 64 | 3.2 | 2 | 0.9 |
| CSNK2A1 | NV298A | Transfection Carrier | C | 1000 | 2.8 | 64 | 2.6 | 5 | 6.7 |
| CDKL3 | NV290A | Transfection Carrier | N | 1000 | 2.2 | 83 | 4.5 | 8 | 2.0 |
| CDKL5 | NV291A | Transfection Carrier | N | 1000 | 4.6 | 84 | 1.3 | 4 | 1.8 |
| JNK3 | NV148A | Transfection Carrier | C | 1000 | 3.1 | 36 | 3.9 | −4 | 0.8 |
| MAPK11 | NV165A | Transfection Carrier | N | 1000 | 5.4 | 35 | 2.3 | 0 | 2.6 |
| MAPK14 | NV166A | Transfection Carrier | C | 1000 | 3.7 | 22 | 1.5 | 0 | 1.7 |
| NLK | NV382A | Transfection Carrier | C | 1000 | 3.2 | 30 | 3.4 | −1 | 3.5 |
| NEK11 | NV377A | Transfection Carrier | N | 1000 | 3.9 | 52 | 4.2 | 7 | 3.6 |
| NEK1 | NV376A | Transfection Carrier | N | 1000 | 5.9 | 38 | 1.7 | 3 | 4.1 |
| NEK2 | NV178A | Transfection Carrier | N | 1000 | 3.4 | 46 | 2.7 | 6 | 6.1 |
| NEK4 | NV378A | Transfection Carrier | N | 1000 | 3.8 | 25 | 0.8 | −12 | 5.6 |
| PAK4 | NV184A | Transfection Carrier | C | 1000 | 11.1 | 25 | 5.5 | 1 | 2.4 |
| MAP4K3 | NV163A | Transfection Carrier | N | 1000 | 7.6 | 50 | 1.4 | 8 | 1.5 |
| STK11 | NV208A | Transfection Carrier | N | 1000 | 3.5 | 81 | 2.3 | −1 | 0.9 |
| SLK | NV205A | Transfection Carrier | N | 1000 | 2.5 | 87 | 3.8 | 36 | 2.9 |
| DAPK2 | NV299A | Transfection Carrier | N | 1000 | 2.5 | 53 | 3.4 | 3 | 1.6 |
| MAP3K2 | NV347A | Transfection Carrier | C | 1000 | 3.2 | 47 | 2.9 | 6 | 1.7 |
| PLK2 | NV408A | Transfection Carrier | N | 1000 | 3.0 | 71 | 3.2 | 4 | 8.5 |
| PLK3 | NV409A | Transfection Carrier | N | 1000 | 3.2 | 52 | 0.8 | 4 | 1.9 |
| PLK4 | NV188A | Transfection Carrier | N | 1000 | 8.6 | 52 | 3.9 | 4 | 1.2 |
| STK35 | NV432A | Transfection Carrier | C | 1000 | 3.4 | 60 | 5.9 | 16 | 3.3 |
| STK17B | NV427A | Transfection Carrier | C | 1000 | 1.9 | 56 | 2.5 | 0 | 3.8 |
| TLK2 | NV444A | Transfection Carrier | C | 1000 | 3.7 | 1 | 3.9 | 0 | 3.2 |
| BRSK2 | NV111A | Transfection Carrier | N | 1000 | 15.9 | 79 | 2.5 | 3 | 2.4 |
| MARK2 | NV172A | Transfection Carrier | N | 1000 | 4.2 | 76 | 1.7 | 4 | 2.1 |
| MELK | NV174A | Transfection Carrier | N | 1000 | 5.8 | 43 | 6.8 | −2 | 2.4 |
| CSNK1A1L | NV295A | Transfection Carrier | N | 1000 | 3.6 | 19 | 4.3 | −6 | 2.9 |
| CSNK1D | NV296A | Transfection Carrier | N | 1000 | 3.5 | 30 | 2.3 | −4 | 1.4 |
| CSNK1G2 | NV118A | Transfection Carrier | N | 1000 | 3.4 | 47 | 1.2 | 1 | 2.8 |
| SIK3 | NV204A | Transfection Carrier | N | 1000 | 12.8 | 62 | 0.8 | 0 | 3.3 |
| SNRK | NV424A | Transfection Carrier | N | 1000 | 4.0 | 68 | 3.7 | −4 | 7.7 |
| CAMK1 | NV253A | Transfection Carrier | N | 1000 | 2.4 | 54 | 2.5 | 7 | 2.6 |
| CAMK2A | NV256A | Transfection Carrier | N | 1000 | 5.8 | 64 | 0.7 | 3 | 2.3 |
| CAMK2D | NV257A | Transfection Carrier | N | 1000 | 5.7 | 68 | 1.3 | 3 | 2.2 |
| CHEK2 | NV293A | Transfection Carrier | C | 1000 | 2.4 | 40 | 4.4 | 0 | 5.0 |
| DCLK3 | NV300A | Transfection Carrier | C | 1000 | 2.4 | 61 | 2.7 | 0 | 3.4 |
| MKNK2 | NV371A | Transfection Carrier | N | 1000 | 2.6 | 64 | 3.0 | 1 | 4.6 |
| PHKG2 | NV388A | Transfection Carrier | N | 1000 | 2.7 | 50 | 1.4 | 3 | 2.5 |
| MAP3K3 | NV349A | Transfection Carrier | C | 1000 | 3.1 | 36 | 3.3 | 4 | 1.9 |
| RIOK2 | NV196A | Transfection Carrier | N | 1000 | 7.1 | 31 | 3.4 | 9 | 6.8 |
| MAP4K5 | NV350A | Transfection Carrier | C | 1000 | 3.2 | 26 | 1.2 | 36 | 4.0 |
| MAST3 | NV353A | Transfection Carrier | N | 1000 | 2.5 | 44 | 8.8 | −1 | 6.6 |
| MAST4 | NV354A | Transfection Carrier | N | 1000 | 2.2 | 46 | 6.0 | 6 | 6.4 |
| STK32B | NV210A | Transfection Carrier | N | 1000 | 3.8 | 18 | 4.3 | −1 | 1.9 |
| STK3 | NV430A | Transfection Carrier | N | 1000 | 3.9 | 43 | 3.5 | 1 | 8.8 |
| STK38 | NV212A | Transfection Carrier | C | 1000 | 6.8 | 24 | 0.5 | 1 | 2.2 |
| STK38L | NV434A | Transfection Carrier | C | 1000 | 3.9 | 20 | 2.1 | 5 | 2.8 |
| PAK6 | NV386A | Transfection Carrier | C | 1000 | 3.3 | 24 | 13.4 | −7 | 23.7 |
| AKT2 | NV103A | Transfection Carrier | C | 1000 | 3.5 | 22 | 1.7 | −1 | 4.7 |
| PKMYT1 | NV187A | Transfection Carrier | C | 1000 | 2.6 | 30 | 1.1 | 6 | 1.7 |
| PRKACA | NV190A | Transfection Carrier | C | 1000 | 6.9 | 56 | 3.1 | −1 | 1.4 |
| PRKACB | NV411A | Transfection Carrier | C | 1000 | 3.6 | 26 | 3.5 | 5 | 3.5 |
| PRKCE | NV412A | Transfection Carrier | C | 1000 | 3.3 | 30 | 8.1 | −6 | 6.1 |
| SGK1 | NV422A | Transfection Carrier | C | 1000 | 3.0 | 43 | 4.5 | −1 | 1.1 |
| WEE2 | NV450A | Transfection Carrier | N | 1000 | 2.8 | 69 | 2.7 | −4 | 2.6 |
| RIPK1 | NV417A | Transfection Carrier | N | 1000 | 2.8 | 25 | 1.8 | 23 | 3.9 |
| RIPK2 | NV197A | Transfection Carrier | N | 1000 | 9.1 | 64 | 1.5 | 43 | 0.5 |
| TNNI3K | NV446A | Transfection Carrier | C | 1000 | 4.0 | 65 | 0.9 | 85 | 1.4 |
| MLTK | NV372A | Transfection Carrier | N | 1000 | 4.4 | 62 | 5.4 | −3 | 8.7 |
| MAP3K12 | NV158A | Transfection Carrier | N | 1000 | 3.7 | 39 | 1.0 | 12 | 6.8 |
| MAP3K19 | NV346A | Transfection Carrier | C | 1000 | 3.0 | 8 | 4.4 | 6 | 5.7 |
| MAP3K21 | NV348A | Transfection Carrier | N | 1000 | 3.2 | 33 | 0.6 | 3 | 5.3 |
| MAP3K4 | NV159A | Transfection Carrier | C | 1000 | 4.8 | 90 | 1.7 | −1 | 2.6 |