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. 2021 Sep 18;26(18):5673. doi: 10.3390/molecules26185673

Table 4.

A new class of α2,3-ST Cst-06 inhibitors (Data from [125]).

#/% Inhibition at 500 μM
First type
graphic file with name molecules-26-05673-i004.jpg graphic file with name molecules-26-05673-i005.jpg
13/51.7 14/58.5
Second type
graphic file with name molecules-26-05673-i006.jpg graphic file with name molecules-26-05673-i007.jpg
15/29.2 16/33.5
graphic file with name molecules-26-05673-i008.jpg
R = H R = (CH2)4NH2 R = (CH2)2CO2H R = (CH2)2CONH2 R = Inline graphic
17/10.5 18/10.7 19/30.5 20/19.1 21/25.1
Third type
graphic file with name molecules-26-05673-i010.jpg
graphic file with name molecules-26-05673-i011.jpg graphic file with name molecules-26-05673-i012.jpg graphic file with name molecules-26-05673-i013.jpg graphic file with name molecules-26-05673-i014.jpg graphic file with name molecules-26-05673-i015.jpg graphic file with name molecules-26-05673-i016.jpg
22/27.2 23/31.7 24/28.0 25/38.1 26/39.5 27/43.1
graphic file with name molecules-26-05673-i017.jpg graphic file with name molecules-26-05673-i018.jpg graphic file with name molecules-26-05673-i019.jpg graphic file with name molecules-26-05673-i020.jpg graphic file with name molecules-26-05673-i021.jpg graphic file with name molecules-26-05673-i022.jpg
28/22.3 29/28.7 30/12.7 31/15.9 32/40.5 33/29.5
graphic file with name molecules-26-05673-i023.jpg graphic file with name molecules-26-05673-i024.jpg graphic file with name molecules-26-05673-i025.jpg graphic file with name molecules-26-05673-i026.jpg graphic file with name molecules-26-05673-i027.jpg graphic file with name molecules-26-05673-i028.jpg
34/78.4 35/79.4 36/9.0 37/50.1 38/27.4 39/33.8