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. 2021 Sep 18;26(18):5673. doi: 10.3390/molecules26185673

Table 5.

Carbamate-linked uridyl-based hST6Gal-I inhibitors (Data from [134]).

Compound # % Inhibition at 10 μM Ki (μM)
graphic file with name molecules-26-05673-i029.jpg
R =
graphic file with name molecules-26-05673-i030.jpg 46 58.9 1.1 ± 0.1
graphic file with name molecules-26-05673-i031.jpg 47 36.6 19.2 ± 2.1
graphic file with name molecules-26-05673-i032.jpg 48 30.9 20.3 ± 2.0
graphic file with name molecules-26-05673-i033.jpg 49 78.0 11.5 ± 5.6
graphic file with name molecules-26-05673-i034.jpg 50 66.4 8.5 ± 1.0