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| assay type | FPPQ | |
|---|---|---|
| solubility [mmol/ml] | 1.4 | |
| microsomal stability [CLint μL/min/mg] | rat | 12.8 |
| human | 8.2 | |
| cytochrome P450 inhibition | 1A2 | 12 μM |
| 2C19 | 10 μM | |
| 3A4 | 57 μM | |
| 2C9 | <25% inh at 10 μM | |
| 2D6 | <25% inh at 10 μM | |
