Table 1. Structure and h-NAAA Inhibitory Activity (IC50) of Compounds 1–15a.
h-NAAA (fluo.), data are expressed as mean ± SD (n ≥ 3).
n.a.: not active @50 μM (<10% inhibition).
h-NAAA (fluo.), data are expressed as mean ± SD (n ≥ 3).
n.a.: not active @50 μM (<10% inhibition).