. 2021 Sep 1;64(18):13327–13355. doi: 10.1021/acs.jmedchem.1c00575

Table 2. Structure and h-NAAA Inhibitory Activity (IC₅₀) of Pyrazole-Substituted Compounds 16–29^a.

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h-NAAA (fluo.), data are expressed as mean ± SD (n ≥ 3).

n.a.: not active @50 μM (<10% inhibition).

Table 2. Structure and h-NAAA Inhibitory Activity (IC50) of Pyrazole-Substituted Compounds 16–29a.