Table 4. h-NAAA Inhibitory Activity (IC50) and LipE Values of Novel Pyrazole-Azabicyclic Sulfonamides 47–50.
h-NAAA (fluo), data are expressed as mean ± SD (n ≥ 3).
LipE = pIC50 – c Log P [c Log P computed using PipelinePilot WebPort 2017] (see also Table S1, Supporting Information).
