. 2020 May 21;5:100083. doi: 10.1016/j.bbih.2020.100083

Table 1.

IC₅₀values of TSPO ligands using [³H] PK 11195 (2 nM final concentration) binding to rat kidney membranes at 4 °C for 90 min in the absence (total binding) or the presence of unlabeled PK 11195, MGV-1, 2-Cl-MGV-1 and 2,4-Di-Cl-MGV-1 at a concentrations ranging from 1 nM to 10 μM.

TSPO ligands	IC₅₀values (nM)
PK 11195	6
MGV-1	350
2-Cl-MGV-1	350
2,4-Di-Cl-MGV-1	100
CB86	1.6
CB204	117.7