TABLE 4.

A list of histone demethylase inhibitors under different phases of clinical trial and their indication.

Histone demethylase inhibitor
Classification	Compounds	Structure	Clinical stage	References
LSD1 inhibitors	Tranylcypromine analogue (GSK2879552)		Clinical	Kalin et al. (2018)
	Bizine		Preclinical	Kim et al. (2020)
	PG11144		Preclinical	Zhu et al. (2012)
		Namoline		Preclinical	Sewry et al. (2019)
	JmjC domain inhibitors	IOX1		Preclinical	Hoyle et al. (2021)
			KDM6B		Preclinical	Basu Mallik et al. (2017)