TABLE 5.
A list of histone deacetylase inhibitors under different phases of clinical trial and their indication.
Histone acetyltransferase inhibitors | ||||
---|---|---|---|---|
Classification | Compounds | Structure | Clinical stage | References |
HDAC1/2i | MRLB-223 |
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Preclinical | Newbold et al. (2013) |
HDAC3i | BG45 |
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Preclinical | Tang et al. (2018) |
HDAC6i | Rocilinostat (ACY-1215) |
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clinical | Yang et al. (2020) |
Tubacin |
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Preclinical | Liang et al. (2019) | |
HDAC8i | C1A |
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Preclinical | Kaliszczak et al. (2013) |
HPOB |
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Preclinical | Liu et al. (2018) | |
PCI-34051 |
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Preclinical | Morgen et al. (2020) | |
C149 |
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Preclinical | Suzuki et al. (2012) |