Table 2.
Percentage of growth inhibition at 24 h of CAS and CAS in combination with H5K1.
| Drug µg/ml | CAS | CAS in combination with: | |||
|---|---|---|---|---|---|
| 0.25 µg/ml H5K1 | 2.5 µg/ml H5K1 | 25 µg/ml H5K1 | 250 µg/ml H5K1 | ||
| 4 | 90.3 | 89.7 | 89.6 | 89.6 | 94.5 |
| 2 | 93.1 | 93.3 | 93.1 | 93.0 | 94.2 |
| 1 | 94.5 | 94.7 | 94.6 | 94.8 | 95.7 |
| 0.5 | 95.8 | 95.7 | 95.9 | 95.8 | 96.1 |
| 0.25 | 90.4 | 94.4 | 96.0 | 95.8 | 96.2 |
| 0.125 | 79.0 | 94.0 | 93.1 | 93.1 | 94.0 |
| 0.0625 | 68.1⁎ | 69.1⁎ | 77.1⁎ | 80.4⁎ | 79.3⁎ |
| 0.03125 | 16.5 | 15.6 | 15.4 | 18.9 | 23.8 |
| 0.0156 | 11.9 | 12.6 | 9.8 | 11.3 | 13.3 |
| 0.0078 | 11.5 | 11.0 | 9.9 | 11.7 | 10.8 |
The MIC50 breakpoints are marked with *.