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. Author manuscript; available in PMC: 2022 Sep 15.
Published in final edited form as: J Am Chem Soc. 2021 Aug 31;143(36):14438–14444. doi: 10.1021/jacs.1c07117

Figure 1.

Figure 1.

(A) Importance of benzylic N-azoles in drug discovery. (B) Impact of regioselectivity of heterocyclic compounds in medicinal chemistry. (C) Copper-catalyzed regioselective cross couplings of benzylic C–H bonds and N–H heterocycles enabled by various additives.