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. 2021 Sep 28;12(20):1980–1991. doi: 10.18632/oncotarget.28079

Table 2. Drug classes of selected small-molecule drugs.

Drug Class
Trametinib MEK1/2 inhibitor
Crizotinib Tyrosine kinase inhibitor
Larotrectinib TRK inhibitor
Selpercatinib RET inhibitor
Vemurafenib BRAF inhibitor
Regorafenib Tyrosine kinase inhibitor
ONC201 Imipridone
ONC206 Imipridone
ONC212 Imipridone
Rucaparib PARP inhibitor
Olaparib PARP inhibitor
Selumetinib MEK inhibitor
Dabrafenib BRAF inhibitor
Dasatinib Tyrosine kinase inhibitor
Duvelisib PI3K inhibitor
9-ING-41 GSK-3 inhibitor

Drug name is listed in the first column and drug class is listed in the second column.