Table 3.
| feed ratio (mg) |
|||||||||
|---|---|---|---|---|---|---|---|---|---|
| no. | scale (mg) | HPMA | MA-GFLG–PTX | MA-Tyr | [CTA]/[I] | Mw (kDa) | PDI | yield (%) | drug% (wt) |
| P-3 | 200 | 156 | 44 | 1.25 | 105 | 1.12 | 81 | 6.6 | |
| P-8 | 1200 | 857 | 327 | 16 | 1.5 | 90.9 | 1.09 | 63 | 6.1 |
| P-16 | 1180 | 937.2 | 244.5 | 1.25 | 118.7 | 1.20 | 68.5 | 6.3 | |
| P-37 | 5000 | 4220 | 780 | 1.25 | 109.8 | 1.27 | 78 | 7.9 | |
DMSO/H2O 3:1 (v/v) as solvent, monomer concentration 16.6% (wt).
VA-044 as initiator, 40 °C for 48 h.
[M]/[CTA] = 1040.