Table 5.
HPMA Copolymer–GEM/PTX Conjugates for Evaluation of Treatment Efficacy
conjugate | Mw (kDa) | PDI | drug (%) | |
---|---|---|---|---|
GEM | mP–GEM300 | 310 | 1.16 | 7.0 |
mP–GEM200 | 218 | 1.12 | 7.4 | |
2P–GEM | 121 | 1.24 | 8.8 | |
P–GEM | 48 | 1.20 | 8.0 | |
PTX | mP–PTX200 | 213 | 1.32 | 7.0 |
2P–PTX | 92 | 1.15 | 7.5 | |
P–PTX | 29 | 1.06 | 7.6 |