Skip to main content
. Author manuscript; available in PMC: 2022 Feb 12.
Published in final edited form as: J Med Chem. 2021 Jul 16;64(15):11045–11062. doi: 10.1021/acs.jmedchem.1c00439

Figure 1.

Figure 1.

Overview of known androgen receptor antagonists. Clinically approved agents include steroidal antiandrogen (1), first-generation (24) second-generation (57) antiandrogens, as well as an indirect androgen synthesis inhibitor (8).