Table 1.

ABCA1 is a Therapeutic Drug Target

Type	Name	Structure	Drug Group	References
	ATP		Investigational, nutraceutical	DrugBank
	Glyburide		Approved
	Probucol		Approved, investigational
	Tocofersolan		Approved
	Vitamin E		Approved, nutraceutical, vet-approved
	Tamoxifen		Approved
Agonist	Metformin		Approved	[92]
	Atorvastatin		Approved	[93]
	Rosuvastatin		Approved	[94]
	T0901317		Animal studies	[95]
	GW3965			[95]
	GW6340			[96]
	IMB-808			[97]
	22(R)-Hydroxycholesterol			[98]
	LXR-623		Investigational	[99]
Antagonist	TPHP		Animal studies	[100]
	EHDPP			[100]
	SR9238			[101,102]
	SR9243			[103,104]
	GSK2033			[104]