Table 2.
List of Amino acids exposed to the Predicted Binding Sites on tiTac3Ra. (refer Figure 2).
| Binding Site | Involved Amino Acid on tiTac3Ra |
|---|---|
| Binding pocket A | Thr12, Asn13, His14, Thr15, Asn16, Gln17, Phe18, Val19, Gln20, Pro22, Ile25, Asn82, Tyr85, Ala86, Ala87, His88, Gly89, Glu90, Trp91, Cys98, His101, Asn102, Pro105, Val106, Val109, Leu158, Ser162, Ile170, Arg173, Ile175, Cys176, Tyr177, Val178, Tyr190, His191, Val194, Thr195, Val198, Tyr199, Trp255, Tyr258, His259, Phe262, Ile277, Gln278, Tyr281, Leu282, Met285, Ala288, Met289. |
| Binding pocket B | Leu64, Leu67, Asp71, Met74, Met116, Val247, Thr250, Phe251, Ser291, Thr292, Tyr294, Asn295, Ile298, Tyr299. |
| Orthosteric Antagonist binding pocket | Asn78, Phe82, His101, Pro105, Val106, Val109, Phe110, Ile175, Tyr177, Val178, Val194, Thr195, Trp255,Tyr258, His259, Phe262, Met285, Ala288, Met289. |