| ADCs | Antibody-drug conjugates |
| mAbs | Monoclonal antibodies |
| bsADCs | Bispecific ADCs |
| BSB | Binding-Site Barrier |
| PRLR | Prolactin receptor |
| GO | Gemtuzumab ozogamicin |
| BV | Brentuximab Vedotin |
| DAR | Drug-to-antibody ratio |
| T-DM1 | Τrastuzumab emtasine |
| AML | Acute myeloid leukemia |
| Val-Cit | Valine-citrulline |
| PABC | Para-amino-benzyloxycarbonyl |
| PBDs | Pyrrolobenzodiazepines |
| TRX | 1,2,4-trioxolane |
| uAA | Unnatural amino-acids |
| mTG | Microbial transglutaminase |
| SortA | Sortase A |
| FGE | Formylglycine-generating enzyme |
| V-ATPase | Vacuolar H+-ATPase |
| CPT | Camptothecin |
| AF-HPA | Auristatin F-hydroxypropylamide |
| MMAE | Monomethyl auristatin E |
| MMAF | Monomethyl auristatin F |
| TM-ADC | Trastuzumab–maytansinoid ADC |
| AAC | Antibody-antibiotic conjugate |
| MRSA | Methicillin-resistant Staphylococcus aureus |
| MSSA | Methicillin-susceptible Staphylococcus aureus |