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. Author manuscript; available in PMC: 2022 Apr 22.
Published in final edited form as: J Med Chem. 2021 Apr 2;64(8):4903–4912. doi: 10.1021/acs.jmedchem.1c00005

Figure 3. Characterization of the kinetics of binding to hMcl-1 by peptide 15 and 16.

Figure 3.

Kinetics measurements for agents 15 (panel A) and 16 (panel B). Percent inhibition were measured using the DELFIA assay at the indicated concentrations and at various time points. Curve fitting of the observed inhibition as function of the compound concentration provided Ki and kinact, as reported.