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. 2021 Oct 20;17:2611–2620. doi: 10.3762/bjoc.17.174

Table 4.

Results of antiproliferative activity testing (IC50 values less than 10 μM are marked with an asterisk, while a dash denotes an IC50 value higher than 100 μM).

compound IC50 (μM), 72 h, MTT test

MCF-7 MDA-MB-231 PC-3 HeLa HT-29 A549 MRC-5

3 1.06* 78.55 8.68* N/Aa
4 14.42 70.64 9.60* 17.73 N/A
7 9.18*
8 43.11 4.25* N/A
11 96.31 26.29 18.16 N/A
12 82.42 11.19 43.71 36.57
13 69.61 16.39
14 6.97* 24.07
15 21.65 23.59 N/A
16 98.90 33.90 43.04 68.07
17 95.91 19.56
18 22.92 22.46 82.60 19.48 27.15 79.75
19 14.79 12.07 34.35 N/A
20 N/A 87.47 61.74
21 37.24 21.67 9.31* 98.50 N/A
22 45.57 6.06*
23 7.60* 11.44 N/A
24 5.18* 12.26 77.61
DOX [53] 0.20* 0.09* 84.23 0.07* 0.15* 4.91* 0.10*

aIC50 value not available due to nonlinear dose dependence or hormetic effect.