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. 2021 Nov 1;4:1241. doi: 10.1038/s42003-021-02772-0

Table 2.

IC50 values for KRAS mRNA knockdown by AZD4785.

Treatment IC50, M
PC9
 Vehicle 1.473*10−7
 Thioperamide 1.631*10−7
 U18666A 0.935*10−7
 Control siRNA 1.516*10−7
 Rab27a siRNA 1.580*10-7
IC50
LK2
 Vehicle 2.836*10−5
 Thioperamide 5.001*10−7
 U18666A 1.933*10−7
 Control siRNA 4.417*10−6
 Rab27a siRNA 2.581*10−6