Table 1.
Cytokine | Receptor | kon (M−1 s−1) | koff (s−1) | KD (nM) |
---|---|---|---|---|
HIL-23 | IL-23R | 3.0 × 104 | 1.2 × 10−3 | 40 |
HIL-23D36K/W37K/T38K | IL-23R | 1.9 × 104 | 1.1 × 10−3 | 57 |
HIL-12 | IL-12Rβ2 | 1.9 × 106 | 1.9 × 10−3 | 0.987 |
HIL-12D36K/W37K/T38K | IL-12Rβ2 | 3.2 × 106 | 2.7 × 10−3 | 0.840 |
SPR analysis of HIL-23 and HIL-12 variants binding to IL-23R-Fc and IL-12Rβ2-Fc. IL-23R-Fc and IL-12Rβ2-Fc were immobilized on a Protein A chip and increasing concentrations of HIL-23 or HIL-12 variants were injected at a flow rate of 30 μl/min. Measurements were carried out on a Biacore X100 instrument.