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. 2021 May 20;137(20):2817–2826. doi: 10.1182/blood.2020007376

Table 3.

AEs leading to discontinuation of prior KI

Intolerant AE on prior tyrosine KI Grade 2 (n) Grade 3 (n) Grade 4 (n) All grades (n)
Rash 6 8 14
Arthralgia 3 5 1 9
Atrial fibrillation 5 2 1 8
Bleeding 1 3 4
Fatigue 2 2 4
Anorexia/weight loss 3 3
Colitis 1 2 3
Congestive heart failure 1 1 1 3
Pneumonitis 2 1 3
Bruising 2 2
Diarrhea 1 1 2
Hypertension 2 2
Nausea 2 2
Cough 1 1
Dizziness 1 1
Edema 1 1
Gastrointestinal toxicity 1 1
Hyperuricemia 1 1
Infection 1 1
Malaise 1 1
Mental status change 1 1
Myalgia 1 1
Pericardial effusion 1 1
Respiratory failure 1 1
Tendonitis 1 1
Brain abscess 1 1
Transaminitis 1 1
TOTAL 39 28 6 73